Drofenine: a 2‐APB analog with improved selectivity for human TRPV3
نویسندگان
چکیده
منابع مشابه
Drofenine: a 2-APB analog with improved selectivity for human TRPV3
Transient receptor potential vanilloid-3 (TRPV3) is a member of the TRPV subfamily of TRP ion channels. The physiological functions of TRPV3 are not fully understood, in part due to a lack of selective agonists and antagonists that could both facilitate the elucidation of roles for TRPV3 in mammalian physiology, as well as potentially serve as therapeutic agents to modulate conditions for which...
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ژورنال
عنوان ژورنال: Pharmacology Research & Perspectives
سال: 2014
ISSN: 2052-1707,2052-1707
DOI: 10.1002/prp2.62